e-Drug3D

1766

PHENMETRAZINE

DISCONTINUED

INN
PHENMETRAZINE

(is an active metabolite)

cas 134-49-6

CLASS

NERVOUS SYSTEM
ANTIANOREXIC
APPETITE DEPRESSANTS
CNS AGENTS
SYMPATHOMIMETICS

ROUTE (list)

ORAL

ATC code

PK parameters

Target

TARGET NORADRENALINE TRANSPORTER
DOPAMINE TRANSPORTER

DrugCentral

Sodium-dependent noradrenaline transporter UNIPROT P23975 SLC6A2

Sodium-dependent dopamine transporter UNIPROT Q01959 SLC6A3

Download SDF file

3-methyl-2-phenylmorpholine

Formula:
C11H15NO

Calculated chemical properties:

MW 177.24
NB_atoms 13
XLogP 1.74
PSA 24.312
NB_HD 1
NB_HA 2
fsp3 0.45
Lipinski(0=no;1=yes) 1

FDA
NDA 010460 (pdf not found) INN (PHENMETRAZINE HYDROCHLORIDE) PRELUDIN (BOEHRINGER INGELHEIM) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 011752 (pdf not found) INN (PHENMETRAZINE HYDROCHLORIDE) PRELUDIN (BOEHRINGER INGELHEIM) APPROVAL= - YEAR= 0 DISCONTINUED