e-Drug3D

1243

SUFENTANIL

INN
SUFENTANIL

cas 56030-54-7

CLASS

NERVOUS SYSTEM
ANALGESIC
ANESTHETICS
NARCOTICS
OPIATE AGONISTS

ROUTE (list)

INJECTION SUBLINGUAL

ATC code

N01AH03

PK parameters

VD 611 LITER (65 KILOGRAM)
Cl 58.5 LITER / HOUR (65 KILOGRAM)
PPB 93 PERCENT
t1/2 2.7 HOUR

Target

TARGET MU-TYPE OPIOID RECEPTOR

DrugCentral

Mu-type opioid receptor UNIPROT P35372 OPRM1

Download SDF file

N-[4-(methoxymethyl)-1-(2-thiophen-2-ylethyl)piperidin-4-yl]-N-phenylpropanamide

Formula:
C22H30N2O2S

Calculated chemical properties:

MW 386.55
NB_atoms 27
XLogP 4.21
PSA 27.396
NB_HD 0
NB_HA 4
fsp3 0.50
Lipinski(0=no;1=yes) 1

FDA
NDA 074406 (pdf not found) INN (SUFENTANIL CITRATE) SUFENTANIL CITRATE (WATSON LABS) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 019050 (label) INN (SUFENTANIL CITRATE) SUFENTA PRESERVATIVE FREE (RISING) APPROVAL= AP YEAR= 1984
NDA 074413 (pdf not found) INN (SUFENTANIL CITRATE) SUFENTANIL CITRATE (HIKMA) APPROVAL= AP YEAR= 1995
NDA 074534 (pdf not found) INN (SUFENTANIL CITRATE) SUFENTANIL CITRATE (HOSPIRA) APPROVAL= AP YEAR= 1996
NDA 209128 (label) INN (SUFENTANIL CITRATE) DSUVIA (VERTICAL PHARMS) APPROVAL= AP YEAR= 2018 DISCONTINUED