e-Drug3D

1232

BETHANIDINE

DISCONTINUED

INN
BETHANIDINE

cas 55-73-2

CLASS

CARDIOVASCULAR
ADRENERGIC AGENTS
ANTIHYPERTENSIVE AGENTS
SYMPATHOLYTICS

ROUTE (list)

ORAL

ATC code

C02CC01

PK parameters

t1/2 39 HOUR (PMID641213)

Target

DrugCentral

Sodium-dependent noradrenaline transporter UNIPROT P23975 SLC6A2

Download SDF file

Guanidine, N,N'-dimethyl-N''-(phenylmethyl)-

Formula:
C10H15N3

Calculated chemical properties:

MW 177.25
NB_atoms 13
XLogP 0.98
PSA 35.15
NB_HD 2
NB_HA 3
fsp3 0.30
Lipinski(0=no;1=yes) 1

FDA
NDA 017675 (pdf not found) INN (BETHANIDINE SULFATE) TENATHAN (ROBINS AH) APPROVAL= AP YEAR= 1981 NEWMOLECULARENTITY DISCONTINUED