e-Drug3D

1217

ACETOPHENAZINE

DISCONTINUED

INN
ACETOPHENAZINE

cas 2751-68-0

CLASS

NERVOUS SYSTEM
ANTIPSYCHOTIC
DOPAMINE RECEPTOR ANTAGONIST

ROUTE (list)

ORAL

ATC code

N05AB07

PK parameters

Target

TARGET D(1A) DOPAMINE RECEPTOR
D(2) DOPAMINE RECEPTOR

D(2) dopamine receptor UNIPROT P14416 DRD2

Download SDF file

1-[10-[3-[4-(2-hydroxyethyl)piperazin-1-yl]propyl]phenothiazin-3-yl]ethanone

Formula:
C23H29N3O2S

Calculated chemical properties:

MW 411.56
NB_atoms 29
XLogP 3.49
PSA 49.368
NB_HD 1
NB_HA 5
fsp3 0.43
Lipinski(0=no;1=yes) 1

FDA
NDA 012254 (pdf not found) INN (ACETOPHENAZINE MALEATE) TINDAL (SCHERING) APPROVAL= AP YEAR= 1961 DISCONTINUED