e-Drug3D

1862

BENZHYDROCODONE

DISCONTINUED

INN
BENZHYDROCODONE

cas 1259440-61-3

CLASS

NERVOUS SYSTEM
ANALGESIC
NARCOTICS
PRODRUG OF HYDROCODONE AND HYDROMORPHONE
CONVERTED TO ACTIVE HYDROCODONE BY ENZYMES IN THE INTESTINAL TRACT

ROUTE (list)

ORAL

PK parameters

Target

TARGET MU-TYPE OPIOID RECEPTOR

Download SDF file

Morphinan-6-ol, 6,7-didehydro-4,5-epoxy-3-methoxy-17-methyl-, 6-benzoate, (5alpha)-

Formula:
C25H25NO4

Calculated chemical properties:

MW 403.46
NB_atoms 30
XLogP 3.72
PSA 50.738
NB_HD 0
NB_HA 5
fsp3 0.40
Lipinski(0=no;1=yes) 1

FDA
NDA 208653 (label) INN (ACETAMINOPHEN ; BENZHYDROCODONE HYDROCHLORIDE) APADAZ (ZEVRA THERAP) APPROVAL= AP YEAR= 2018 DISCONTINUED