e-Drug3D

1549

M FESOTERODINE

INN
FESOTERODINE

cas 207679-81-0

CLASS

ANTISPASMODICS
ANTIMUSCARINIC
MUSCARINIC ANTAGONIST
OVERACTIVE BLADDER WITH SYMPTOMS OF URGE URINARY INCONTINENCE
URINARY ANTISPASMODICS
GENITO
HYDROLYSIS BY NONSPECIFIC ESTERASES

ROUTE (list)

ATC code

G04BD11

PK parameters

F 52 PERCENT
Tmax 1.8 HOUR
Cmax 11.6 NANOMOLAR (8 MILLIGRAM)
VD 169 LITER
Cl 13.6 LITER / HOUR (EQN)
PPB 50 PERCENT
t1/2 8.59 HOUR

Target

TARGET MUSCARINIC RECEPTOR

DrugCentral

Muscarinic acetylcholine receptor M2 UNIPROT P08172 CHRM2

Muscarinic acetylcholine receptor M3 UNIPROT P20309 CHRM3

Download SDF file

Benzenemethanol, 3-[(1R)-3-[bis(1-methylethyl)amino]-1-phenylpropyl]-4-hydroxy-

Formula:
C22H31NO2

Calculated chemical properties:

MW 341.48
NB_atoms 25
XLogP 4.53
PSA 46.686
NB_HD 2
NB_HA 3
fsp3 0.45
Lipinski(0=no;1=yes) 1

FDA
-